Last update : 11.07.2025
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Cotrina, E.Y., Santos, L.M., Rivas, J., Blasi, D., Leite, J.P., Liz, M.A., Busquets, M.A., Planas, A., Prohens, R., Gimeno, A., Jiménez-Barbero, J., Gales, L., Llop, J., Quintana, J., Cardoso, I., Arsequell, G. "Targeting transthyretin in Alzheimer's disease: Drug discovery of small-molecule chaperones as disease-modifying drug candidates for Alzheimer's disease" European Journal of Medicinal Chemistry., 226: art.n° 113847. (2021).
Light, T.P., Brun, D., Guardado-Calvo, P., Pederzoli, R., Haouz, A., Neipel, F., Rey, F.A., Hristova, K., Backovic, M. "Human herpesvirus 8 molecular mimicry of ephrin ligands facilitates cell entry and triggers EphA2 signaling" PloS Biology., 19(9): art.n° e3001392. (2021).
Scholl, D., Sigoillot, M., Overtus, M., Colomer Martinez, R., Martens, C., Wang, Y., Pardon, E., Laeremans, T., Garcia-Pino, A., Steyaert, J., Sheppard, D.N., Hendrix, J., Govaerts, C. "A topological switch in CFTR modulates channel activity and sensitivity to unfolding" Nature Chemical Biology., 17(9): 989–997. (2021).
Carivenc, C., Maveyraud, L., Blanger, C., Ballereau, S., Roy-Camille, C., Nguyen, M.C., Génisson, Y., Guilhot, C., Chalut, C., Pedelacq, J.D., Mourey, L. "Phosphopantetheinyl transferase binding and inhibition by amidino-urea and hydroxypyrimidinethione compounds" Scientific Reports., 11: art.n° 18042. (2021).
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Song, L., Merceron, R., Hulpia, F., Lucía, A., Gracia, B., Jian, Y., Risseeuw, M.D.P., Verstraelen, T., Cos, P., Aínsa, J.A., Boshoff, H.I.M., Munier-Lehmann, H., Savvides, S.N., Van Calenbergh, S. "Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors" European Journal of Medicinal Chemistry., 225: art.n° 113784. (2021).
Muller, M.C., Wagner, T. "The Oxoglutarate Binding Site and Regulatory Mechanism Are Conserved in Ammonium Transporter Inhibitors GlnKs from Methanococcales" International Journal of Molecular Sciences., 22(16): art.n° 8631. (2021).