PUBLICATIONS
- Vantieghem, T., Osipov, E.M., Beelen, S., Strelkov, S.V. "Crystal engineering of the hepatoma-derived growth factor-related protein 2 PWWP domain towards crystallographic fragment screening" Acta Crystallographica F., 81(8): 358-364. (2025).
- Kalandia, G., Declerck, K., Salazar Marcano, D.E., Gourmand, R., Moussawi, M.A., Parac-Vogt, T.N. "Finding the Key: Binding of Metal-Oxo Clusters to the Enzyme Active Site Enabled by “Click” (Bio)Conjugation" Angewandte Chemie International Edition., 64(50): art.n° e202518349. (2025).
- Gerusz, V., Regenass, P., Rousseau, Q., Moraine, V., Justine Dao, J., Xavier Lavé, X., Das, S., Hue Perron, J., Fajas Descamps, L., Bravo, J., Dieppois, G., Kaplan, N., Lefebre, M., Altomari, D., Romanov, V., Finn, T., Daram, P., Bernardini, F., Gross, M., Lysek, R., Adam, A., Pohin, D., Maio, M., Tatsis, V., Sunose, M., Ronin, C., Ciesielski, F., Ahlstrand, J., Jacobsson, S., Unemo, M., Cameron, D.R "The bactericidal FabI inhibitor Debio 1453 clears antibiotic-resistant Neisseria gonorrhoeae infection in vivo" nature Communications., 16: art.n° 8309 . (2025).
- Sarmadi, F., Caza, A., Gao, Z., Rochel, N., Gleason, J.L., White, J.H. "Hyperagonism of a Vitamin D Receptor Agonist/Histone Deacetylase Inhibitor Hybrid Molecule" Journal of Medicinal Chemistry., 68(19): 20675-20688. (2025).
- Wehbi, H., Cece, Q., Phan, G., Broutin, I. "MexB/inhibitor complexes preparation for crystallography and cryo-EM, comparison and possible pitfalls" Methods in Enzymology., 724: 365-396. (2025).
- Zampieri, V., Vermot, A., Thepaut, M., Petit-Hartlein I., Fieschi, F., Falson, P., Chaptal, V. "X-ray diffraction images for two membrane protein crystals presenting high anisotropy; the B. subtilis ABC transporter BmrA and the S. pneumoniae NADPH oxidase" IUCr Data., 10(7): art.n° x250591. (2025).
- Kyrko, D., Cao, T., Retailleau, P., Kaffy, J., Crousse, B. "Access to N-Fluorinated Azapeptides and Azapeptoids as Peptidomimetic Scaffolds" ACS Organic & Inorganic Au., 5(6): 531–538. (2025).
- Vieira Da Cruz, A., Perraudin, V., Minopoli, N., Iacono, R., Roig-Zamboni, V., Bossio, A., Tangara, S., Fayolle, M., Kanazawa, A., Philouze, C., Tarallo, A., Heming, J.J.A., Artola, M., Behr, J.B., Overkleeft, H.S., Moracci, M., Sulzenbacher, G., Parenti, G., Py, S. "C-Branched Iminosugars as Selective Pharmacological Chaperones of Lysosomal α-Glucosidase for the Treatment of Pompe Disease" Journal of Medicinal Chemistry., 68(18): 19269–19286. (2025).
- Song, Z.Y., Zhang, X., Ai, X., Huang, L.Y., Hou, X.M., Fossé, P., Liu, N.N., Mauffret, O., Réty, S., Xi, X.G. "Structural mechanism of RECQ1 helicase in unfolding G-quadruplexes compared with duplex DNA" Nucleic Acids Research., 53(17): art.n° gkaf877. (2025).
- De Colibus, L., Ludzi, P., Biasutto, A., Pica, A., Hopper, J.T.S., Jazayeri, A., Dürr, K.L. "Improved structure of mouse gasdermin D: a new blueprint for structure-based drug design" Acta Crystallographica F., 81(10): 408-415. (2025).