PUBLICATIONS
- Kuki, Walmsley, D.L., Kanai, K., Takechi, S., Yoshida, M., Murakami, R., Takano, K., Tominaga, Y., Takahashi, M., Ito, S., Nakao, N., Angove, H., Baker, L.M., Carter, E., Dokurno, P., Le Strat, L., Macias, A.T., Molyneaux, C.A., Murray, J.B., Surgenor, A.E., Hamada, T., Hubbard, R.E. "A covalent fragment-based strategy targeting a novel cysteine to inhibit activity of mutant EGFR kinase". RSC Medicinal Chemistry, 14(12):2731-2737. (2023).
- Cornelius, P., Mayes, B.A., Petersen, J.S., Turnquist, D.J., Dufour, P.J., Dannenberg, A.J., Shanahan, J.M., Carver, B.J. "Pharmacological Characterization of SDX-7320/Evexomostat: A Novel Methionine Aminopeptidase Type 2 Inhibitor with Anti-tumor and Anti-metastatic Activity ". Molecular Cancer Therapeutics, 23(5):595–605. (2024).
- Contaldo, U., Santucci, P., Vergnes, A., Leone, P., Becam, J., Biaso, F., Ilbert, M., Ezraty, B., Lojou, E., Mazurenko, I. "How the Larger Methionine-Rich Domain of CueO from Hafnia alvei Enhances Cuprous Oxidation" JACS Au., 5(4): 1833-1844. (2025).
- Panek, D., Pasieka, A., Jończyk,J., Gawlińska,M., Zaręba,P., Siwek,A., Wolak,M., Mordyl,B., Głuch-Lutwin,M., Latacz,G., Brazzolotto,X., Chantegreil,F., Nachon,F., Karasova, J.Z., Pejchal, J., Mzik, M., Sestak, V., Prchal, L., Odvarkova, J., Soukup, O., Korabecny, J., Sorf, A., Hamsikova, M., Zemanova, L., Muckova, L., Vánova, N., Dryja, P., Sałat,K., Höfner, G., Wanner, K., Więckowska,A., Malawska, B. "Multifunctional, Fluorene-Based Modulator of Cholinergic and GABAergic Neurotransmission as a Novel Drug Candidate for Palliative Treatment of Alzheimer's Disease" Angewandte Chemie International Edition., 64(6): art.n° e202420510. (2025).
- Danis, C., Dupré, E., Bouillet, T., Denéchaud, M., Lefebvre, C., Nguyen, M., Mortelecque, J., Cantrelle, F.X., Rain, J.C., Hanoulle, X., Colin, M., Buée, L., Landrieu, I. "Inhibition of tau neuronal internalization using anti-tau single domain antibodies" Nature Communications., 16: art.n° 3162. (2025).
- Malard, F., Dias, K., Baudy, M., Thore, S., Vialet, B., Barthélémy, B., Fribourg, S., Karginov, F.V., Campagne, S. "Molecular basis for the calcium-dependent activation of the ribonuclease EndoU" Nature Communications., 16: art.n° 3110. (2025).
- Liao, J., Hameed, U.F.S., Hoffmann, T.D., Kurze, E., Sun, G., Steinchen, W., Nicoli, A., Di Pizio, A., Kuttler, C., Song, C., Catici, D.A.M., Assaad-Gerbert, F., Hoffmann, T., Arold, S.T., Schwab, W.G. "β-Carotene alleviates substrate inhibition caused by asymmetric cooperativity" Nature Communications., 16: art.n° 3065. (2025).
- Hladík, P., Brunoni, F., Žukauskaitė,A., Zatloukal,M., Bělíček,J., Kopečný, D., Briozzo, P., Ferchaud, N., Novák, O., Pěnčík, A. "Phenylacetic acid metabolism in land plants: novel pathways and metabolites" Journal of Experimental Botany., 76(12): 3427–3443. (2025).
- Ewert, W., Bartens, C., Ongouta, J., Holmes, M., Heutling, A., Kishore, A., Urbansky, T., Zeilinger, C., Preller, M., Kirschning, A. "Structure and function of the geldanamycin amide synthase from Streptomyces hygroscopicus" Nature Communications., 16: art.n° 2464. (2025).
- Karlsson, E., Andén, O., Fan, C., Fourati, Z., Haouz, A., Zhuang, Y., Howard, R.J., Delarue, M., Lindahl, E. "Vestibular modulation by stimulant derivatives in a pentameric ligand-gated ion channel" British Journal of Pharmacology., 182(12): 2790-2802. (2025).