RECHERCHER
Résultats de la recherche ""
Optimal Stapling of a Helical Peptide-Foldamer Hybrid Using a C-terminal 4-Mercaptoproline Enhances Protein Surface Recognition and Cellular Activity
Publié le 28/02/2025
... Neuville, M., Bourgeais, M., Buratto, J., Saragaglia, C., Li, B., Galeano-Otero, I., Mauran, L., Varajao, L., Goudreau, S.R., Kauffmann, B., Thinon, E., Pasco, M., Khatib, A.M., Guichard, G. "Optimal Stapling of a Helical Peptide-Foldamer Hybrid Using a C ...
Structural Plasticity of Flavin-Dependent Thymidylate Synthase Controlled by the Enzyme Redox State
Publié le 25/02/2025
... Pecqueur, L., Lombard, M., Hamdane, D. "Structural Plasticity of Flavin-Dependent Thymidylate Synthase Controlled by the Enzyme Redox State" Biomolecules., 15(3): art.n° 318. (2025). ...
Unraveling the molecular grammar and the structural transitions underlying the fibrillation of a viral fibrillogenic domain
Publié le 25/02/2025
... Gondelaud, F., Leval, J., Arora, L., Walimbe, A., Bignon, C., Ptchelkine, D., Brocca, S., Mukhopadyay, S., Longhi, S. "Unraveling the molecular grammar and the structural transitions underlying the fibrillation of a viral fibrillogenic domain" Protein ...
Identification of ß-Glucocerebrosidase Activators for Glucosylceramide hydrolysis
Publié le 22/02/2025
... Schulze, M.S.E.D., Scholz, D., Jnoff, E., Hall, A., Melin, J., Sands, Z.A., Rodriguez, E., Andre, V.M. "Identification of ß-Glucocerebrosidase Activators for Glucosylceramide hydrolysis" ChemMedChem., 19(7): art.n° e202300548. (2024). ...
Novel, tightly structurally related N-myristoyltransferase inhibitors display equally potent yet distinct inhibitory mechanisms
Publié le 22/02/2025
... Rivière, F., Dian, C., Dutheil, R.F., Monassa, P., Giglione, C., Meinnel, T. "Novel, tightly structurally related N-myristoyltransferase inhibitors display equally potent yet distinct inhibitory mechanisms" Structure., 32(10): 1737-1750. (2024). ...
ATP mimetics targeting prolyl-tRNA synthetases as a new avenue for antimalarial drug development
Publié le 22/02/2025
... Mishra, S., Malhotra, N., Laleu, B., Chakraborti, S., Yogavel, M., Sharma, A. "ATP mimetics targeting prolyl-tRNA synthetases as a new avenue for antimalarial drug development" iScience., 27(7): art.n° 110049. (2024). ...
Discovery, Optimization, and Biological Evaluation of Arylpyridones as Cbl-b Inhibitors
Publié le 22/02/2025
... Mfuh, A.M., Boerth, J.A., Bommakanti, G., Chan, C., Chinn, A.J., Code, E., Fricke, P.J., Giblin, K.A., Gohlke, A., Hansel, C., Hariparsad, N., Hughes, S.J., Jin, M., Kantae, V., Kavanagh, S.L., Lamb, M.L., Lane, J., Moore, R., Puri, T., Quinn, T.R., Reddy ...
Mechanistic and Structural Insights on Difluoromethyl-1,3,4-oxadiazole Inhibitors of HDAC6.
Publié le 22/02/2025
... Cellupica, E., Gaiassi, A., Rocchio, I., Rovelli, G., Pomarico, R., Sandrone, G., Caprini, G., Cordella, P., Cukier, C., Fossati, G., Marchini, M., Bebel, A., Airoldi, C., Palmioli, A., Stevenazzi, A., Steinkuhler, C., Vergani, B. "Mechanistic and ...
Cucurbituril-like Giant PolyOxoThiometalate: Structural Analysis and Solution Studies
Publié le 18/02/2025
... Marrot, J., Falaise, C., Abou Fadel, M., Leclerc, N., Haouas, M., Floquet, S., Sécheresse, F., Cadot, E. "Cucurbituril-like Giant PolyOxoThiometalate: Structural Analysis and Solution Studies" Inorganic Chemistry., 64(8): 4017–4024. (2025). ...
The Soap Opera of Metal Catalysis in Epoxy-Acid Vitrimers
Publié le 18/02/2025
... Ciardi, D., Retailleau, I., Tournilhac, F. "The Soap Opera of Metal Catalysis in Epoxy-Acid Vitrimers" Macromolecules., 58(7): 3377–3385. (2025). ...