RECHERCHER
Résultats de la recherche ""
Structural Plasticity of Flavin-Dependent Thymidylate Synthase Controlled by the Enzyme Redox State
Publié le 25/02/2025
... Pecqueur, L., Lombard, M., Hamdane, D. "Structural Plasticity of Flavin-Dependent Thymidylate Synthase Controlled by the Enzyme Redox State" Biomolecules., 15(3): art.n° 318. (2025). ...
Identification of ß-Glucocerebrosidase Activators for Glucosylceramide hydrolysis
Publié le 22/02/2025
... Schulze, M.S.E.D., Scholz, D., Jnoff, E., Hall, A., Melin, J., Sands, Z.A., Rodriguez, E., Andre, V.M. "Identification of ß-Glucocerebrosidase Activators for Glucosylceramide hydrolysis" ChemMedChem., 19(7): art.n° e202300548. (2024). ...
Novel, tightly structurally related N-myristoyltransferase inhibitors display equally potent yet distinct inhibitory mechanisms
Publié le 22/02/2025
... Rivière, F., Dian, C., Dutheil, R.F., Monassa, P., Giglione, C., Meinnel, T. "Novel, tightly structurally related N-myristoyltransferase inhibitors display equally potent yet distinct inhibitory mechanisms" Structure., 32(10): 1737-1750. (2024). ...
ATP mimetics targeting prolyl-tRNA synthetases as a new avenue for antimalarial drug development
Publié le 22/02/2025
... Mishra, S., Malhotra, N., Laleu, B., Chakraborti, S., Yogavel, M., Sharma, A. "ATP mimetics targeting prolyl-tRNA synthetases as a new avenue for antimalarial drug development" iScience., 27(7): art.n° 110049. (2024). ...
Discovery, Optimization, and Biological Evaluation of Arylpyridones as Cbl-b Inhibitors
Publié le 22/02/2025
... Mfuh, A.M., Boerth, J.A., Bommakanti, G., Chan, C., Chinn, A.J., Code, E., Fricke, P.J., Giblin, K.A., Gohlke, A., Hansel, C., Hariparsad, N., Hughes, S.J., Jin, M., Kantae, V., Kavanagh, S.L., Lamb, M.L., Lane, J., Moore, R., Puri, T., Quinn, T.R., Reddy ...
Mechanistic and Structural Insights on Difluoromethyl-1,3,4-oxadiazole Inhibitors of HDAC6.
Publié le 22/02/2025
... Cellupica, E., Gaiassi, A., Rocchio, I., Rovelli, G., Pomarico, R., Sandrone, G., Caprini, G., Cordella, P., Cukier, C., Fossati, G., Marchini, M., Bebel, A., Airoldi, C., Palmioli, A., Stevenazzi, A., Steinkuhler, C., Vergani, B. "Mechanistic and ...
Structural insights into tecovirimat antiviral activity and poxvirus resistance
Publié le 14/02/2025
... Vernuccio, R., Martínez León, A., Poojari, C.S., Buchrieser, J., Selverian, C.N., Jaleta, Y., Meola, A., Guivel-Benhassine, F., Porrot, F., Haouz, A., Chevreuil, M., Raynal, B., Mercer, J., Simon-Loriere, S., Chandran, K., Schwartz, O., Hub, J.S., ...
Charge Transfer Between Ce and Fe During Cooling of an Aluminosilicate Melt: An In Situ XANES Investigation
Publié le 11/02/2025
... Donatini, A., Georges, P., Fevre, T., Cormier, L., Neuville, D.R. "Charge Transfer Between Ce and Fe During Cooling of an Aluminosilicate Melt: An In Situ XANES Investigation" Inorganic Chemistry., 64(7): 3528–3540. (2025). ...
Structure predictions of MuRF1-UBE2 complexes identify amino acid residues governing interaction selectivity for each MuRF1-E2 pair
Publié le 11/02/2025
... Claustre, A., Malige, M., Macheton, M., Combaret, L., Lefai, E., Fafournoux, P., Taillandier, D., Henri, J., Polge, C. "Structure predictions of MuRF1-UBE2 complexes identify amino acid residues governing interaction selectivity for each MuRF1-E2 pair" ...
RING dimerisation drives higher-order organisation of SINA/SIAH E3 ubiquitin ligases
Publié le 07/02/2025
... Coste, F., Mishra, A., Chapuis, C., Mance, L., Pukało,Z., Bigot,N., Goffinont, S., Gaudon, V., Garnier, N., Talhaoui, I., Castaing, B., Huet, S., Suskiewicz, M.J. "RING dimerisation drives higher-order organisation of SINA/SIAH E3 ubiquitin ligases" FEBS ...