RECHERCHER
Résultats de la recherche ""
Human herpesvirus 8 molecular mimicry of ephrin ligands facilitates cell entry and triggers EphA2 signaling
Publié le 15/09/2021
... Light, T.P., Brun, D., Guardado-Calvo, P., Pederzoli, R., Haouz, A., Neipel, F., Rey, F.A., Hristova, K., Backovic, M. "Human herpesvirus 8 molecular mimicry of ephrin ligands facilitates cell entry and triggers EphA2 signaling" PloS Biology., 19(9): art ...
Targeting transthyretin in Alzheimer's disease: Drug discovery of small-molecule chaperones as disease-modifying drug candidates for Alzheimer's disease
Publié le 15/09/2021
... Cotrina, E.Y., Santos, L.M., Rivas, J., Blasi, D., Leite, J.P., Liz, M.A., Busquets, M.A., Planas, A., Prohens, R., Gimeno, A., Jiménez-Barbero, J., Gales, L., Llop, J., Quintana, J., Cardoso, I., Arsequell, G. "Targeting transthyretin in Alzheimer's ...
Development and crystallography-aided SAR studies of multifunctional BuChE inhibitors and 5-HT6R antagonists with β-amyloid anti-aggregation properties
Publié le 14/09/2021
... Wichur, T., Godyń,J., Góral,I., Latacz,G., Bucki,A., Siwek,A., Głuch-Lutwin,M., Mordyl,B., Śniecikowska,J., Walczak,M., Knez,D., Jukic,M., Sałat,K., Gobec,S., Kołaczkowski,M., Malawska,B., Brazzolotto,X., Więckowska, A. "Development and crystallography ...
Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors
Publié le 14/09/2021
... Song, L., Merceron, R., Hulpia, F., Lucía, A., Gracia, B., Jian, Y., Risseeuw, M.D.P., Verstraelen, T., Cos, P., Aínsa, J.A., Boshoff, H.I.M., Munier-Lehmann, H., Savvides, S.N., Van Calenbergh, S. "Structure-aided optimization of non-nucleoside M. ...
Nonhydrolysable Analogues of (p)ppGpp and (p)ppApp Alarmone Nucleotides as Novel Molecular Tools
Publié le 14/09/2021
... Mojr, V., Roghanian, M., Tamman, H., Pham, D.D.D., Petrová, M., Pohl, R., Takada, H., Van Nerom, K., Ainelo, H., Caballero-Montes, J., Jimmy, S., Garcia-Pino, A., Hauryliuk, V., Rejman, D. "Nonhydrolysable Analogues of (p)ppGpp and (p)ppApp Alarmone ...
Estimation of stress in specimens loaded with ultrasonic fatigue machines
Publié le 14/09/2021
... Jacquemain, V., Ranc, N., Cheuleu, C., Michel, V., Favier, V., Castelnau, O., Vinci, D., Thiaudiere, D., Mocuta, C. "Estimation of stress in specimens loaded with ultrasonic fatigue machines" International Journal of Fatigue., 153: art.n° 106474. (2021). ...
Exploring the dNTP -binding site of HIV-1 reverse transcriptase for inhibitor design
Publié le 14/09/2021
... Gu, W., Martinez, S., Singh, A.K., Nguyen, H., Rozenski, J., Schols, D., Herdewijn, P., Das, K., De Jonghe, S. "Exploring the dNTP -binding site of HIV-1 reverse transcriptase for inhibitor design" European Journal of Medicinal Chemistry., 225: art.n° ...
Crystal structures capture multiple stoichiometric states of an aqueous self-assembling oligourea foldamer
Publié le 14/09/2021
... Collie, G.W., Lombardo, C.M., Yoo, S.Y., Pułka-Ziach, C., Gabelica, V., MacKereth, C.D., Rosu, F., Guichard, G. "Crystal structures capture multiple stoichiometric states of an aqueous self-assembling oligourea foldamer" Chemical Communications., 57(75): ...
Phosphopantetheinyl transferase binding and inhibition by amidino-urea and hydroxypyrimidinethione compounds
Publié le 14/09/2021
... Carivenc, C., Maveyraud, L., Blanger, C., Ballereau, S., Roy-Camille, C., Nguyen, M.C., Génisson, Y., Guilhot, C., Chalut, C., Pedelacq, J.D., Mourey, L. "Phosphopantetheinyl transferase binding and inhibition by amidino-urea and hydroxypyrimidinethione ...
The Oxoglutarate Binding Site and Regulatory Mechanism Are Conserved in Ammonium Transporter Inhibitors GlnKs from Methanococcales
Publié le 13/08/2021
... Muller, M.C., Wagner, T. "The Oxoglutarate Binding Site and Regulatory Mechanism Are Conserved in Ammonium Transporter Inhibitors GlnKs from Methanococcales" International Journal of Molecular Sciences., 22(16): art.n° 8631. (2021). ...