Dernière mise à jour : 07/11/2025
Ong, S.T., Bajaj, S., Tanner, M.R., Chang, S.C., Krishnarjuna, B., Ng, X.R., Morales, R.A.V., Chen, M.W., Luo, D., Patel, D.J., Yasmin, S., Ng, J.J.H., Zhuang, Z., Nguyen, H.M., El Sahili, A., Lescar, J., Patil, R., Charman, S.A., Robins, E.G., Coggi, J., Tan, P.W., Sadasivam, P., Ramasamy, B., Hartimath, S.V., Dhawan, V., Bednenko, J., Colussi, P., Wulff, H., Pennington, M.W., Kuyucak, S., Norton, R.S., Beeton, C., Chandy, G. "Modulation of lymphocyte potassium channel KV1.3 by membrane-penetrating, joint-targeting immunomodulatory plant defensin" ACS Pharmacology & Translational Science., 3(4): 720–736. (2020).
Tamman, H., Van Nerom, K., Takada, H., Vandenberk, N., Scholl, D., Polikanov, Y., Hofkens, J., Talavera, A., Hauryliuk, V., Hendrix, J., Garcia-Pino, A. "A nucleotide-switch mechanism mediates opposing catalytic activities of Rel enzymes" Nature Chemical Biology., 16(8): 834–840. (2020).
Ahmad, L., Plancqueel, S., Lazar, N., Korri-Youssoufi, H., Li de la Sierra-Gallay, I., van Tilbeurgh, H., Salmon, L. "Novel N-substituted 5-phosphate-d-arabinonamide derivatives as strong inhibitors of phosphoglucose isomerases: synthesis, structure-activity relationship and crystallographic studies" Bioorganic Chemistry., 102: art.n° 104048. (2020).
Dietrich, C., Li de la Sierra‐Gallay, I., Masi, M., Girard, E., Dautin, N., Constantinesco‐Becker, F., Tropis, M., Daffé, M., van Tilbeurgh, H., Bayan, N. "The C‐terminal domain of Corynebacterium glutamicum mycoloyltransferase A is composed of five repeated motifs involved in cell wall binding and stability" Molecular Microbiology., 114(1): 1-16. (2020).
Mori, M., Stelitano, G., Gelain, A., Pini, E., Chiarelli, L.R., Sammartino, J.C., Poli, G., Tuccinardi, T., Beretta, G., Porta, A., Bellinzoni, M., Villa, S., Meneghetti, F. "Shedding X-ray light on the role of magnesium in the activity of M. tuberculosis salicylate synthase (MbtI) for drug design" Journal of Medicinal Chemistry., 63(13): 7066–7080. (2020).
Fourati, Z., Sauguet, L., Delarue, M. "Structural evidence for the binding of monocarboxylates and dicarboxylates at pharmacologically relevant extracellular sites of a pentameric ligand-gated ion channel" Acta Crystallographica D., 76(7): 668-675. (2020).
Sosa Fajardo, A., Legrand, P., Payá-Tormo, L., Martin, L., Pellicer Martinez, M.T., Echavarri-Erasun, C., Vernède, X., Rubio, L.M., Nicolet, Y. "Structural insights into the mechanism of the radical SAM carbide synthase NifB, a key nitrogenase cofactor maturating enzyme" Journal of the American Chemical Society., 142(25): 11006–11012. (2020).
McPhillie, M.J., Zhou, Y., Hickman, M.R., Gordon, J.A., Weber, C.R., Li, Q., Lee, P.J., Amporndanai, K., Johnson, R.M., Darby, H., Woods, S., Li, Z., Priestley, R.S., Ristroph, K.D., Biering, S.B., El Bissati, K., Hwang, S., Esaa Hakim, F., Dovgin, S.M., Lykins, J.D., Roberts, L., Hargrave, K., Cong, H., Sinai, A.P., Muench, S.P., Dubey, J.P., Prud'homme, R.K., Lorenzi, H.A., Biagini, G.A., Moreno, S.N., Roberts, C.W., Antonyuk, S.V., Fishwick, C.W.G., McLeod, R. "Potent Tetrahydroquinolone Eliminates Apicomplexan Parasites" Frontiers in Cellular and Infection Microbiology., 10: art.n° 203. (2020).
Charenton, C., Gaudon Plesse, C., Back, R., Ulryck, N., Cosson, L., Séraphin, B., Graille, M. "Pby1 is a direct partner of the Dcp2 decapping enzyme" Nucleic Acids Research., 48(11): 6353–6366. (2020).
Machtens, D.A., Willerding, J.M., Eschenburg, S., Reubold, T.F. "Crystal structure of the metaeffector MesI (Lpg2505) from Legionella pneumophila" Biochemical and Biophysical Research Communications., 527(3): 696-701. (2020).