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Publications

Dernière mise à jour : 07/11/2025
E.g., 07/11/2025
E.g., 07/11/2025
Kiyeleko, S., Hocine, S., Mautino, G., Kuenemann, M., Nawrotek, A., Miallau, L., Vuillard, L.M., Mirguet, O., Kotschy, A., Hanessian, S. "Targeting non-alcoholic fatty liver disease: Design, X-ray co-crystal structure and synthesis of ‘first-in-kind’ inhibitors of serine/threonine kinase25" Bioorganic & Medicinal Chemistry Letters., 75: art.n° 128950. (2022).
Bermeo, R., Lal, K., Ruggeri, D., Lanaro, D., Mazzotta, S., Vasile, F., Imberty, A., Belvisi, L., Varrot, A., Bernardi, A. "Targeting a Multidrug-Resistant Pathogen: First Generation Antagonists of Burkholderia cenocepacia’s BC2L-C Lectin" ACS Chemical Biology., 17(10): 2899–2910. (2022).
Seoane, S., Gogoi, P., Zárate-Ruíz, A., Peluso-Iltis, C., Peters, S., Guiberteau, T., Maestro, M.A., Pérez-Fernández, R., Rochel, N., Mouriño, A. "Design, Synthesis, Biological Activity, and Structural Analysis of Novel Des-C-Ring and Aromatic-D-Ring Analogues of 1α,25-Dihydroxyvitamin D3" Journal of Medicinal Chemistry., 65(19): 13112-13124. (2022).
Roovers, M., Labar, G., Wolff, P., Feller, A., Van Elder, D., Soin, R., Gueydan, C., Kruys, V., Droogmans, L. "The Bacillus subtilis open reading frame ysgA encodes the SPOUT methyltransferase RlmP forming 2’-O-methylguanosine at position 2553 in the A-loop of 23S rRNA." RNA., 28(10): 1185-1196. (2022).
Yoo, S.H., Buratto, J., Roy, A., Morvan, E., Pasco, M., Pulka-Ziach, K., Lombardo, C.M., Rosu, F., Gabelica, V., Mackereth, C.D., Collie, G.W., Guichard, G. "Adaptive Binding of Alkyl Glycosides by Nonpeptidic Helix Bundles in Water: Toward Artificial Glycolipid Binding Proteins" Journal of the American Chemical Society., 144(35): 15988–15998. (2022).
Fadel, F., Bassim, V., Francis, V.I., Porter, S.L., Botzanowski, T., Legrand, P., Maté Perez, M., Bourne, Y., Cianférani, S., Vincent, F. "Insights into the atypical autokinase activity of the Pseudomonas aeruginosa GacS histidine kinase and its interaction with RetS" Structure., 30(9): 1285-1297. (2022).
Iannelli, G., Milite, C., Marechal, N., Cura, V., Bonnefond, L., Troffer-Charlier, N., Feoli, A., Rescigno, D., Wang, Y., Cipriano, A., Viviano, M., Bedford, M.T., Cavarelli, J., Castellano, S., Sbardella, G. "Turning Nonselective Inhibitors of Type I Protein Arginine Methyltransferases into Potent and Selective Inhibitors of Protein Arginine Methyltransferase 4 through a Deconstruction–Reconstruction and Fragment-Growing Approach" Journal of Medicinal Chemistry., 65(17): 11574–11606. (2022).
Deflandre, B., Jadot, C., Planckaert, S., Thiébaut, N., Stulanovic, N., Herman, R., Devreese, B., Kerff, F., Rigali, S. "Structure and Function of BcpE2, the Most Promiscuous GH3-Family Glucose Scavenging Beta-Glucosidase" mBio., 13(4): art.n° e00935-22. (2022).
Gogl, G., Zambo, B., Kostmann, C., Cousido-Siah, A., Morlet, B., Durbesson, F., Negroni, L., Eberling, P., Jané, P., Nominé, Y., Zeke, A., Østergaard, S., Monsellier, E., Vincentelli, R., Travé, G. "Quantitative fragmentomics allow affinity mapping of interactomes" Nature Communications., 13: art.n° 5472. (2022).
Notova, S., Bonnardel , F., Rosato, F., Siukstaite, L., Schwaiger, J., Lim, J.H., Bovin, N., Varrot, A., Ogawa, Y., Römer, W., Lisacek, F., Imberty, A. "The choanoflagellate pore-forming lectin SaroL-1 punches holes in cancer cells by targeting the tumor-related glycosphingolipid Gb3" Communications Biology., 5: art.n° 954. (2022).