Last update : 11.07.2025
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Nandwani, N., Bhowmik, D., Glaser, C., Childers, M.C., Goluguri, R.R., Dawood, A., Regnier, M., Houdusse, A., Spudich, J.A., Ruppel, K.M. "Hypertrophic cardiomyopathy mutations Y115H and E497D disrupt the folded-back state of human β-cardiac myosin allosterically" Nature Communications., 16: art.n° 8751. (2025).
Martinkus, J., Terradot, L., Jurėnas, D., Cascales, E. "Widespread deployment of the human CD38 ADP-ribosyl cyclase fold in antibacterial and anti-eukaryotic polymorphic toxins" Journal of Biological Chemistry., 301(11): art.n° 110775. (2025).
Vieira Da Cruz, A., Perraudin, V., Minopoli, N., Iacono, R., Roig-Zamboni, V., Bossio, A., Tangara, S., Fayolle, M., Kanazawa, A., Philouze, C., Tarallo, A., Heming, J.J.A., Artola, M., Behr, J.B., Overkleeft, H.S., Moracci, M., Sulzenbacher, G., Parenti, G., Py, S. "C-Branched Iminosugars as Selective Pharmacological Chaperones of Lysosomal α-Glucosidase for the Treatment of Pompe Disease" Journal of Medicinal Chemistry., 68(18): 19269–19286. (2025).
Moussawi, M.A., Abdelhameed, S.A.M., de Azambuja, F., Wijten, A., Vasović, T., Ćirković Veličković, T., Parac-Vogt, T.N. "Fast and selective protein modification with ironsubstituted polyoxometalates via a radical pathway". Inorganic Chemistry Frontiers., on line first (26/09/2025): (2025).
Vantieghem, T., Osipov, E.M., Beelen, S., Strelkov, S.V. "Crystal engineering of the hepatoma-derived growth factor-related protein 2 PWWP domain towards crystallographic fragment screening" Acta Crystallographica F., 81(8): 358-364. (2025).
De Colibus, L., Ludzi, P., Biasutto, A., Pica, A., Hopper, J.T.S., Jazayeri, A., Dürr, K.L. "Improved structure of mouse gasdermin D: a new blueprint for structure-based drug design" Acta Crystallographica F., 81(10): 408-415. (2025).
Kalandia, G., Declerck, K., Salazar Marcano, D.E., Gourmand, R., Moussawi, M.A., Parac-Vogt, T.N. "Finding the Key: Binding of Metal-Oxo Clusters to the Enzyme Active Site Enabled by “Click” (Bio)Conjugation". Angewandte Chemie International Edition., on line first (25/09/2025): (2025).
Gerusz, V., Regenass, P., Rousseau, Q., Moraine, V., Justine Dao, J., Xavier Lavé, X., Das, S., Hue Perron, J., Fajas Descamps, L., Bravo, J., Dieppois, G., Kaplan, N., Lefebre, M., Altomari, D., Romanov, V., Finn, T., Daram, P., Bernardini, F., Gross, M., Lysek, R., Adam, A., Pohin, D., Maio, M., Tatsis, V., Sunose, M., Ronin, C., Ciesielski, F., Ahlstrand, J., Jacobsson, S., Unemo, M., Cameron, D.R "The bactericidal FabI inhibitor Debio 1453 clears antibiotic-resistant Neisseria gonorrhoeae infection in vivo" nature Communications., 16: art.n° 8309 . (2025).